发明名称 |
GlyT2 modulators |
摘要 |
Certain alpha-, beta-, and gamma-amino acid derivatives are disclosed as selective GlyT2 inhibitors for the treatment of central nervous system (CNS) conditions such as muscle spasticity, tinnitus, epilepsy and neuropathic pain.
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申请公布号 |
US2005119245(A1) |
申请公布日期 |
2005.06.02 |
申请号 |
US20040976067 |
申请日期 |
2004.10.28 |
申请人 |
BARCLAY TRISTIN K.;SANTILLAN ALEJANDRO JR.;TANG LIU Y.;VENKATESAN HARIHARAN;WOLIN RONALD L. |
发明人 |
BARCLAY TRISTIN K.;SANTILLAN ALEJANDRO JR.;TANG LIU Y.;VENKATESAN HARIHARAN;WOLIN RONALD L. |
分类号 |
C07C275/28;C07C275/36;C07C279/28;C07D213/56;C07D277/30;C07D295/13;C07D333/20;C07D333/24;C07K5/06;(IPC1-7):A61K31/55;A61K31/454;A61K31/443;A61K31/426;A61K31/421;A61K31/381;A61K31/165 |
主分类号 |
C07C275/28 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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