发明名称 BENZYLETHER AMINE COMPOUNDS USEFUL AS CCR-5 ANTAGONISTS
摘要 <p>The present invention relates to compounds which are CCR-5 receptor antagonists of the general formula (I) wherein R&lt;1&gt;, R&lt;2&gt;, R&lt;3&gt;, R&lt;4&gt;, R&lt;a&gt;, R&lt;b&gt;, R&lt;c&gt;, R&lt;d&gt;, X, m and n are as defined herein. The invention further comprises pharmaceutical compositions comprising such compounds, as well as the use of such compounds to treat CCR-5 mediated disorders.</p>
申请公布号 WO2005047249(A1) 申请公布日期 2005.05.26
申请号 WO2004US37258 申请日期 2004.11.08
申请人 SCHERING AKTIENGESELLSCHAFT;DAVEY, DAVID;LEE, WHEESEONG;LU, SHOU-FU;PHILLIPS, GARY;WEI, GUO, PING;YE, BIN 发明人 DAVEY, DAVID;LEE, WHEESEONG;LU, SHOU-FU;PHILLIPS, GARY;WEI, GUO, PING;YE, BIN
分类号 A61K31/435;A61K31/135;A61K31/165;A61K31/40;C07C217/58;C07C235/42;C07C255/54;C07C275/28;C07D207/08;C07D207/12;C07D207/14;C07D207/16;C07D211/14;C07D211/26;C07D211/38;C07D211/42;C07D211/44;C07D211/46;C07D211/48;C07D211/52;C07D211/58;C07D211/62;C07D211/64;C07D211/66;C07D213/20;C07D213/30;C07D213/40;C07D213/53;C07D213/64;C07D213/82;C07D213/89;C07D217/06;C07D233/54;C07D233/88;C07D235/26;C07D241/08;C07D295/13;C07D295/192;C07D295/215;C07D295/26;C07D319/08;C07D333/34;C07D401/06;C07D401/12;C07D403/12;C07D405/12;C07D471/10;C07D487/08;C07D491/10;(IPC1-7):C07D207/14 主分类号 A61K31/435
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