发明名称 |
RAPIDLY SOLUBLE DRUG COMPOSITION COMPRISING MICRONIZED AS-3201 |
摘要 |
<p>A fast-dissolving pharmaceutical composition comprising micronized (R)-2-(4-bromo-2-fluorobenzyl)-1,2,3,4-tetrahydropyrroloÄ1,2-aÜpyrazin e-4-spiro-3'-pyrrolidine-1,2',3,5'-tetrone (hereinafter, referred to as AS-3201). The present pharmaceutical composition has improved dissolution characteristics as well as a good bioavailability.</p> |
申请公布号 |
EP1033132(B1) |
申请公布日期 |
2005.05.25 |
申请号 |
EP19980947883 |
申请日期 |
1998.10.15 |
申请人 |
DAINIPPON PHARMACEUTICAL CO., LTD. |
发明人 |
OHASHI, MAMORU;OGASAWARA, KAZUYOSHI;SHIRAI, YOSHIMI;FUJIOKA, HIROSHI |
分类号 |
A61K9/20;A61K31/4985;A61K31/499;A61K47/02;A61K47/12;A61K47/24;A61P3/10;(IPC1-7):A61K31/495 |
主分类号 |
A61K9/20 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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