发明名称 SUBSTITUTED PIPERAZINES, (1,4)DIASZEPINES, AND 2,5-DIAZABICYCLO (2.2.1) HEPTANES AS HISTAMINE H1 AND/OR H3 ANTAGONISTS OR HISTAMINE H3 REVERSE ANTAGONISTS
摘要 The present invention relates to novel piperazine and azepine derivatives having pharmacological activity, processes for their preparation, to compositions containing them and to their use in the treatment of neurodegenerative disorders including Alzheimer's disease.
申请公布号 KR20050049553(A) 申请公布日期 2005.05.25
申请号 KR20057006621 申请日期 2005.04.15
申请人 GLAXO GROUP LIMITED 发明人 ANCLIFF, RACHAEL;ELDRED, COLIN, DAVID;FOGDEN, YVONNE, C;HANCOCK, ASHLEY, PAUL;HEIGHTMAN, THOMAS, DANIEL;HOBBS, HEATHER;HODGSON, SIMON, TEANBY;LINDON, MATTHEW, J;WILSON, DAVID, MATTHEW
分类号 A61P11/00;A61P25/00;C07D209/42;C07D211/46;C07D213/50;C07D213/64;C07D213/81;C07D215/40;C07D215/46;C07D215/50;C07D239/28;C07D243/08;C07D265/36;C07D277/62;C07D285/06;C07D295/092;C07D295/185;C07D295/192;C07D295/215;C07D295/26;C07D307/79;C07D307/85;C07D311/84;C07D317/68;C07D333/38;C07D405/06;C07D487/08;C07D491/04;(IPC1-7):C07D295/192;C07D295/18;C07D401/12 主分类号 A61P11/00
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