发明名称 |
Monocyclic and bicyclic lactams as factor Xa inhibitors |
摘要 |
The present application describes monocyclic and bicyclic lactams and derivatives thereof of Formulae Ia-e: wherein one of one of T<SUP>1 </SUP>and T<SUP>2 </SUP>is carbonyl, thiocarbonyl, or sulfonyl or pharmaceutically acceptable salt forms thereof. Compounds of the present invention are useful as inhibitors of trypsin-like serine proteases, specifically factor Xa.
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申请公布号 |
US2005107361(A1) |
申请公布日期 |
2005.05.19 |
申请号 |
US20040952397 |
申请日期 |
2004.09.28 |
申请人 |
HAN WEI;QIAO JENNIFER X.;HU ZILUN |
发明人 |
HAN WEI;QIAO JENNIFER X.;HU ZILUN |
分类号 |
A61K;A61K31/4709;A61K31/498;A61K31/502;A61K31/538;A61K31/55;(IPC1-7):A61K31/55;A61K31/470;C07D43/02 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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