发明名称 |
SUBSTITUTED 2-PYRIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES |
摘要 |
The invention relates to 3-ketoester of formula (IV) €ƒ€ƒ€ƒ
wherein R1 represents a 2, 3 or 4-pyridine ring optionally substituted by a C 3-6 cycloalkyl group, a C 1-4 alkyl group, a C 1-4 alkoxy group, a benzyl group or a halogen atom, R5 is an halogen atom and R is an alkyl. |
申请公布号 |
PL370349(A1) |
申请公布日期 |
2005.05.16 |
申请号 |
PL20020370349 |
申请日期 |
2002.09.19 |
申请人 |
SANOFI-AVENTIS;MITSUBISHI PHARMA CORP. |
发明人 |
GALLET THIERRY;LARDENOIS PATRICK;LOCHEAD ALISTAIR;MARGUERIE SEVERINE;NEDELEC ALAIN;SAADY MOURAD;SLOWINSKI FRANCK;YAICHE PHILIPPE |
分类号 |
A61K31/519;A61P3/04;A61P3/10;A61P9/10;A61P17/14;A61P25/00;A61P25/02;A61P25/08;A61P25/16;A61P25/18;A61P25/24;A61P25/28;A61P27/02;A61P27/06;A61P35/00;A61P43/00;C07D213/50;C07D213/60;C07D487/04 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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