发明名称 SUBSTITUTED 2-PYRIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-A]PYRIMIDIN-4-ONE AND 7-PYRIDINYL-2,3-DIHYDROIMIDAZO[1,2-A]PYRIMIDIN-5(1H)ONE DERIVATIVES
摘要 The invention relates to 3-ketoester of formula (IV) €ƒ€ƒ€ƒ wherein R1 represents a 2, 3 or 4-pyridine ring optionally substituted by a C 3-6 cycloalkyl group, a C 1-4 alkyl group, a C 1-4 alkoxy group, a benzyl group or a halogen atom, R5 is an halogen atom and R is an alkyl.
申请公布号 PL370349(A1) 申请公布日期 2005.05.16
申请号 PL20020370349 申请日期 2002.09.19
申请人 SANOFI-AVENTIS;MITSUBISHI PHARMA CORP. 发明人 GALLET THIERRY;LARDENOIS PATRICK;LOCHEAD ALISTAIR;MARGUERIE SEVERINE;NEDELEC ALAIN;SAADY MOURAD;SLOWINSKI FRANCK;YAICHE PHILIPPE
分类号 A61K31/519;A61P3/04;A61P3/10;A61P9/10;A61P17/14;A61P25/00;A61P25/02;A61P25/08;A61P25/16;A61P25/18;A61P25/24;A61P25/28;A61P27/02;A61P27/06;A61P35/00;A61P43/00;C07D213/50;C07D213/60;C07D487/04 主分类号 A61K31/519
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