发明名称 COMPOUNDS AND METHODS FOR TREATMENT OF THROMBOSIS
摘要 The present invention provides compounds that inhibit Factor XIa and methods of preventing or treating undesired thrombosis by administering a compound of the invention to a mammal. The invention also provides three-dimensional structures of Factor XIa and methods for designing or selecting additional Factor XIa inhibitors using these structures.
申请公布号 WO2004103270(A3) 申请公布日期 2005.05.12
申请号 WO2004US10349 申请日期 2004.04.02
申请人 SUNTORY PHARMACEUTICAL RESEARCH LABORATORIES LLC;ABDEL-MEGUID, SHERIN, S.;BABINE, ROBERT, E.;DENG, HONGFENG;JIN, LEI;LIN, JIAN;MAGEE, SCOTT, R.;MEYERS, HAROLD, V.;PANDEY, PRAMOD;RYNKIEWICZ, MICHAEL, J.;WEAVER, DAVID, T. 发明人 ABDEL-MEGUID, SHERIN, S.;BABINE, ROBERT, E.;DENG, HONGFENG;JIN, LEI;LIN, JIAN;MAGEE, SCOTT, R.;MEYERS, HAROLD, V.;PANDEY, PRAMOD;RYNKIEWICZ, MICHAEL, J.;WEAVER, DAVID, T.
分类号 A61K;A61K38/00;A61K38/04;C07K2/00;C07K5/04;C07K5/06;C07K5/065;C07K5/078 主分类号 A61K
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