发明名称 NAPHTHALENE-1,5-DISULFONIC ACID SALTS OF A SUBSTITUTED 4-AMINO-1-(PYRIDYLMETHYL)PIPERIDINE COMPOUND
摘要 This invention provides naphthalene-1,5-disulfonic acid salts of 4-{N-[7-(3-(S)-1-carbamoyl-1,1-diphenylmethyl)pyrrolidin-1-yl)hept-1-yl]-N-(isopropyl)amino}-1-(4-methoxypyrid-3-ylmethyl)piperidine, which salts are useful as muscarinic receptor antagonists. This invention is also directed to pharmaceutical compositions comprising these salt forms, methods of using these salt forms for treating medical conditions mediated by muscarinic receptors; and processes for preparing these salt forms.
申请公布号 WO2005042514(A2) 申请公布日期 2005.05.12
申请号 WO2004US35941 申请日期 2004.10.28
申请人 THERAVANCE, INC.;WILSON, RICHARD, D.;CONGDON, JULIE;MAMMEN, MATHAI;ZHANG, WEIJIANG;CHAO, ROBERT 发明人 WILSON, RICHARD, D.;CONGDON, JULIE;MAMMEN, MATHAI;ZHANG, WEIJIANG;CHAO, ROBERT
分类号 A61K31/444;A61K31/4545;C07C309/35;C07D401/14 主分类号 A61K31/444
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