发明名称 ИНГИБИТОРЫ КАТЕПСИН-ЦИСТЕИНПРОТЕАЗЫ
摘要 This invention relates to a novel class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, such as osteoporosis.
申请公布号 RU2004129587(A) 申请公布日期 2005.05.10
申请号 RU20040129587 申请日期 2003.02.28
申请人 МЕРК ФРОССТ КЭНАДА ЭНД КО. (CA);ЭКСИС ФАРМАСЬЮТИКАЛЗ, ИНК. (US) 发明人 БЭЙЛИ Кристофер И. (CA);БЛЭК Кэмерон (CA);ЛЕЖЕ Серж (CA);ЛИ Чун Синг (CA);МАККЭЙ Дэн (CA);МЕЛЛОН Кристоф (CA);ГОТЬЕ Жак Ив (CA);ЛАУ Чеук (CA);ТЕРЬЕН Мишель (CA);ТРУОНГ Воуй-Линх (CA);ГРИН Майкл Дж. (US);ХИРШБЕЙН Бернард Л. (US);ДЖЭНК Джеймс У. (US);ПАЛМЕР Джеймс Т. (US);БАСКАРАН Читра (US)
分类号 C07D295/12;A61K31/275;A61K31/381;A61K31/404;A61K31/417;A61K31/42;A61K31/4245;A61K31/426;A61K31/427;A61K31/44;A61K31/4406;A61K31/4409;A61K31/4465;A61K31/47;A61K31/495;A61K31/505;A61K31/5375;A61K45/00;A61P1/02;A61P3/14;A61P19/02;A61P19/08;A61P19/10;A61P29/00;A61P35/00;A61P43/00;C07C255/25;C07C255/29;C07C255/46;C07C255/58;C07C255/60;C07C259/10;C07C311/37;C07C317/32;C07C317/36;C07D209/08;C07D211/26;C07D211/38;C07D213/36;C07D213/38;C07D213/57;C07D213/61;C07D213/64;C07D213/70;C07D213/71;C07D213/74;C07D213/89;C07D215/12;C07D231/12;C07D233/54;C07D233/64;C07D239/06;C07D239/26;C07D241/12;C07D261/08;C07D263/32;C07D271/06;C07D277/28;C07D295/135;C07D295/22;C07D307/52;C07D333/20;C07D401/04;C07D417/04 主分类号 C07D295/12
代理机构 代理人
主权项
地址