发明名称 |
ИНГИБИТОРЫ КАТЕПСИН-ЦИСТЕИНПРОТЕАЗЫ |
摘要 |
This invention relates to a novel class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, such as osteoporosis. |
申请公布号 |
RU2004129587(A) |
申请公布日期 |
2005.05.10 |
申请号 |
RU20040129587 |
申请日期 |
2003.02.28 |
申请人 |
МЕРК ФРОССТ КЭНАДА ЭНД КО. (CA);ЭКСИС ФАРМАСЬЮТИКАЛЗ, ИНК. (US) |
发明人 |
БЭЙЛИ Кристофер И. (CA);БЛЭК Кэмерон (CA);ЛЕЖЕ Серж (CA);ЛИ Чун Синг (CA);МАККЭЙ Дэн (CA);МЕЛЛОН Кристоф (CA);ГОТЬЕ Жак Ив (CA);ЛАУ Чеук (CA);ТЕРЬЕН Мишель (CA);ТРУОНГ Воуй-Линх (CA);ГРИН Майкл Дж. (US);ХИРШБЕЙН Бернард Л. (US);ДЖЭНК Джеймс У. (US);ПАЛМЕР Джеймс Т. (US);БАСКАРАН Читра (US) |
分类号 |
C07D295/12;A61K31/275;A61K31/381;A61K31/404;A61K31/417;A61K31/42;A61K31/4245;A61K31/426;A61K31/427;A61K31/44;A61K31/4406;A61K31/4409;A61K31/4465;A61K31/47;A61K31/495;A61K31/505;A61K31/5375;A61K45/00;A61P1/02;A61P3/14;A61P19/02;A61P19/08;A61P19/10;A61P29/00;A61P35/00;A61P43/00;C07C255/25;C07C255/29;C07C255/46;C07C255/58;C07C255/60;C07C259/10;C07C311/37;C07C317/32;C07C317/36;C07D209/08;C07D211/26;C07D211/38;C07D213/36;C07D213/38;C07D213/57;C07D213/61;C07D213/64;C07D213/70;C07D213/71;C07D213/74;C07D213/89;C07D215/12;C07D231/12;C07D233/54;C07D233/64;C07D239/06;C07D239/26;C07D241/12;C07D261/08;C07D263/32;C07D271/06;C07D277/28;C07D295/135;C07D295/22;C07D307/52;C07D333/20;C07D401/04;C07D417/04 |
主分类号 |
C07D295/12 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|