发明名称 ARYLAMINE-SUBSTITUTED QUINAZOLINONE COMPOUNDS
摘要 Compounds represented by Formula (I) which are useful as are alpha-1A/B adrenoceptor antagonists, to methods of treating conditions associated with the activity of alpha-1A/B adrenoceptors, and to methods of making said compounds, wherein Ar, Z, R, R', R<5> and R<10> are as defined herein.
申请公布号 WO2005005395(A3) 申请公布日期 2005.05.06
申请号 WO2004EP06973 申请日期 2004.06.28
申请人 F. HOFFMANN-LA ROCHE AG;CONNOLLY, TERRENCE, JOSEPH;KEITZ, PAUL, FRANCIS;LEE, EUN, KYUNG;LI, JIM;LOPEZ-TAPIA, FRANCISCO, JAVIER;MCGARRY, PATRICK, FINBAR;MELVILLE, CHRIS, RICHARD;NITZAN, DOV;O'YANG, COUNDE;PADILLA, FERNANDO;WEINHARDT, KLAUS, KURT 发明人 CONNOLLY, TERRENCE, JOSEPH;KEITZ, PAUL, FRANCIS;LEE, EUN, KYUNG;LI, JIM;LOPEZ-TAPIA, FRANCISCO, JAVIER;MCGARRY, PATRICK, FINBAR;MELVILLE, CHRIS, RICHARD;NITZAN, DOV;O'YANG, COUNDE;PADILLA, FERNANDO;WEINHARDT, KLAUS, KURT
分类号 A61K31/517;A61K31/549;C07D239/90;C07D239/95;C07D285/24;C07D285/26;C07D401/12;C07D401/14;C07D403/12;C07D405/12;C07D413/12;C07D417/02;C07D417/12 主分类号 A61K31/517
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