发明名称 IMIDAZOPYRAZINE TYROSINE KINASE INHIBITORS
摘要 Compounds of the formula (I) and pharmaceutically acceptable salts thereof, wherein Q<1 >and R<1> are defined herein, inhibit the IGF-1R enzyme and are useful for the treatment and/or prevention of various diseases and conditions that respond to treatment by inhibition of tyrosine kinases.
申请公布号 WO2005037836(A2) 申请公布日期 2005.04.28
申请号 WO2004US34219 申请日期 2004.10.14
申请人 OSI PHARMACEUTICALS, INC.;BECK, PATRICIA, ANNE;CESARIO, CARA;COX, MATTHEW;DONG, HAN-QING;FOREMAN, KENNETH;MULVIHILL, MARK, JOSEPH;NIGRO, ANTHONY, INNOCENZO;SAROGLOU, LYDIA;STEINIG, ARNO, G.;SUN, YINGCHUAN;WENG, QINGHUA;WERNER, DOUGLAS;WILKES, ROBIN;WILLIAMS, JONATHAN 发明人 BECK, PATRICIA, ANNE;CESARIO, CARA;COX, MATTHEW;DONG, HAN-QING;FOREMAN, KENNETH;MULVIHILL, MARK, JOSEPH;NIGRO, ANTHONY, INNOCENZO;SAROGLOU, LYDIA;STEINIG, ARNO, G.;SUN, YINGCHUAN;WENG, QINGHUA;WERNER, DOUGLAS;WILKES, ROBIN;WILLIAMS, JONATHAN
分类号 A61K31/4985;C07D487/04 主分类号 A61K31/4985
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