发明名称 NOVEL SOLID BODY FORMS OF MESOPROGESTIN 11beta-[4E-(HYDROXYIMINOMETHYL)-PHENYL]-17alpha-METHOXYMETHYL-17beta-METHOXY-ESTRA-4,9-DIEN-3-ONE
摘要 The invention relates to novel solid body forms of mesoprogestin 11beta-[4E-(hydroxyiminomethyl)-phenyl]-17alpha-methoxymethyl-17beta-methoxy-estra-4,9-dien-3-one (oxime J 867), particularly a highly pure and stable amorphous or highly crystalline form (ansolvate/anhydrate) of compound J 867. The invention also relates to methods for producing said novel solid body forms and to the use thereof in pharmaceutical compositions. The novel solid body forms are characterized by exhibiting a high degree of stability. The solid body forms of oxime J 867 can, in particular, be used in the area of fertility control and in hormone replacement therapy.
申请公布号 EA005623(B1) 申请公布日期 2005.04.28
申请号 EA20020001192 申请日期 2001.05.09
申请人 SCHERING AKTIENGESELLSCHAFT 发明人 GRAWE, DETLEF;HOZEL, PETER;MULLER, UWE;WINTER, GABRIELE
分类号 A61K31/569;A61K31/565;A61P5/36;A61P15/08;A61P15/12;A61P15/18;C07J41/00;(IPC1-7):C07J41/00 主分类号 A61K31/569
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