发明名称 Androgen receptor antagonists
摘要 The present invention is directed to a new class of 6-sulfonamido-quinolin-2-one and 6-sulfonamido-2-oxo-chromene derivatives to their use as androgen antagonists, and to relieve conditions associated with inappropriate activation of the androgen receptor.
申请公布号 US2005085466(A1) 申请公布日期 2005.04.21
申请号 US20040758581 申请日期 2004.01.15
申请人 DU DANIEL Y.;FYFE MATTHEW C.T.;PROCTER MARTIN J.;SCHOFIELD KAREN L.;SHAH VILASBEN K.;WILLIAMS GEOFFREY M. 发明人 DU DANIEL Y.;FYFE MATTHEW C.T.;PROCTER MARTIN J.;SCHOFIELD KAREN L.;SHAH VILASBEN K.;WILLIAMS GEOFFREY M.
分类号 A61K31/452;A61K31/4709;A61K31/496;A61K31/5377;A61K31/541;C07D215/22;C07D215/227;C07D311/54;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D413/02;C07D417/02;C07D417/12;C07D491/08;C07D491/10;(IPC1-7):A61K31/541;A61K31/537;A61K31/470;C07D43/02 主分类号 A61K31/452
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