发明名称 INHIBITORS OF CATHEPSIN S
摘要 The present invention provides compounds, compositions and methods for the selective inhibition of cathepsin S. In a preferred aspect, cathepsin S is selectively inhibited in the presence of at least one other cathepsin isozyme. The present invention also provides methods for treating a disease state in a subject by selectively inhibiting cathepsin S.
申请公布号 WO2005034848(A2) 申请公布日期 2005.04.21
申请号 WO2004US26986 申请日期 2004.08.19
申请人 IRM LLC;LIU, HONG;CHATTERJEE, ARNAB;TULLY, DAVID, C.;ALPER, PHILLIP, B.;BURSULAYA, BADRY;GUO, JIANHUA;WOODMANSEE, DAVID;MUTNICK, DANIEL;KARANEWSKY, DONALD, S.;HE, YUN 发明人 LIU, HONG;CHATTERJEE, ARNAB;TULLY, DAVID, C.;ALPER, PHILLIP, B.;BURSULAYA, BADRY;GUO, JIANHUA;WOODMANSEE, DAVID;MUTNICK, DANIEL;KARANEWSKY, DONALD, S.;HE, YUN
分类号 A61K;A61K31/397;A61K31/401;A61K31/404;A61K31/423;A61K31/445;A61K31/454;A61K31/495;A61K31/537;A61K31/5375;A61K31/54;C07D209/04;C07D209/08;C07D261/14;C07D265/30;C07D295/13;C07D295/18;C07D295/20;C07D411/12;C07D413/12;C07D417/12 主分类号 A61K
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