发明名称 |
DIHYDRONAPHTHALINDERIVATE UND VERFAHREN ZUR HERSTELLUNG DERSELBEN |
摘要 |
Dihydronaphthalene compounds have excellent 17 alpha -hydroxylase/C17-20-lyase inhibiting activity, thromboxan A2 synthesis inhibiting activity, and aromatase inhibiting activity and are thereby are useful as preventive and/or therapeutic agents for various male sex hormone- and female sex hormone-dependent diseases such as prostate cancer, prostatomegaly, masculinization, breast cancer, mastopathy, uterine cancer, endometriosis, and ovarian cancer, as well as myocardial infarction, angina pectoris, and bronchial asthma. |
申请公布号 |
DE69823222(T2) |
申请公布日期 |
2005.04.14 |
申请号 |
DE1998623222T |
申请日期 |
1998.10.01 |
申请人 |
DAIICHI PHARMACEUTICAL CO., LTD. |
发明人 |
HARTMANN, WOLFGANG;WACHALL, BERTIL;YOSHIHAMA, MAKOTO;NAKAKOSHI, MASAMICHI;NOMOTO, SHIN;IKEDA, YOSHIKAZU |
分类号 |
A61K;A61K31/025;A61K31/415;A61K31/4164;A61K31/435;A61K31/44;A61K31/4409;A61P5/24;C07C;C07C13/48;C07C39/225;C07C39/23;C07C43/20;C07C43/21;C07D;C07D213/16;C07D213/24;C07D213/44;C07D233/54;C07D233/64 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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