发明名称 DIHYDRONAPHTHALINDERIVATE UND VERFAHREN ZUR HERSTELLUNG DERSELBEN
摘要 Dihydronaphthalene compounds have excellent 17 alpha -hydroxylase/C17-20-lyase inhibiting activity, thromboxan A2 synthesis inhibiting activity, and aromatase inhibiting activity and are thereby are useful as preventive and/or therapeutic agents for various male sex hormone- and female sex hormone-dependent diseases such as prostate cancer, prostatomegaly, masculinization, breast cancer, mastopathy, uterine cancer, endometriosis, and ovarian cancer, as well as myocardial infarction, angina pectoris, and bronchial asthma.
申请公布号 DE69823222(T2) 申请公布日期 2005.04.14
申请号 DE1998623222T 申请日期 1998.10.01
申请人 DAIICHI PHARMACEUTICAL CO., LTD. 发明人 HARTMANN, WOLFGANG;WACHALL, BERTIL;YOSHIHAMA, MAKOTO;NAKAKOSHI, MASAMICHI;NOMOTO, SHIN;IKEDA, YOSHIKAZU
分类号 A61K;A61K31/025;A61K31/415;A61K31/4164;A61K31/435;A61K31/44;A61K31/4409;A61P5/24;C07C;C07C13/48;C07C39/225;C07C39/23;C07C43/20;C07C43/21;C07D;C07D213/16;C07D213/24;C07D213/44;C07D233/54;C07D233/64 主分类号 A61K
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