发明名称 AMIDE TYPE CARBOXAMIDE DERIVATIVE
摘要 <p>An amide type carboxamide derivative represented by the general formula [1]: [Chemical formula 1] (wherein X represents -N= or -CH=; R&lt;1&gt; represents halogeno, lower alkyl, etc.; R&lt;2&gt; represents, e.g., [Chemical formula 2] Y&lt;1&gt; and Y&lt;2&gt; are the same or different and each represents halogeno or a group selected among lower alkyls, lower alkoxys, etc.; and ring A represents phenyl, etc.) or a pharmacologically acceptable salt of the derivative. The derivative and salt are useful as a medicine, especially an FXa inhibitor.</p>
申请公布号 WO2005030706(A1) 申请公布日期 2005.04.07
申请号 WO2004JP13892 申请日期 2004.09.24
申请人 TANABE SEIYAKU CO., LTD.;KAWAGUCHI, TAKAYUKI;AKATSUKA, HIDENORI;MORIMOTO, MASAMICHI;WATANABE, TATSUYA;IIJIMA, TORU;MURAKAMI, JUN 发明人 KAWAGUCHI, TAKAYUKI;AKATSUKA, HIDENORI;MORIMOTO, MASAMICHI;WATANABE, TATSUYA;IIJIMA, TORU;MURAKAMI, JUN
分类号 A61P7/02;A61P43/00;C07C237/42;C07D409/12;(IPC1-7):C07C237/42;C07D213/81;C07D213/75;C07D265/32;C07D333/40;A61K31/537;A61K31/44;A61K31/422;A61K31/415;A61K31/402;A61K31/381;C07D495/04;C07D413/12;C07D403/14;C07D401/12;C07D401/14 主分类号 A61P7/02
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