发明名称 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO
摘要 <p>Compounds of Formula (IA), IB), IC), and (ID) wherein R<1>, R<2>, R<3>, R<4>, R<5>, and R<6> are as respectively defined herein for Formula (IA), (IB), (IC), and (ID), or a tautomer, prodrug, solvate, or salt thereof; pharmaceutical compositions containing such compounds, and methods of modulating the glucocorticoid receptor function and methods of treating disease-states or conditions mediated by the glucocorticoid receptor function or characterized by inflammatory, allergic, or proliferative processes in a patient using these compounds.</p>
申请公布号 WO2005030213(A1) 申请公布日期 2005.04.07
申请号 WO2004US31009 申请日期 2004.09.22
申请人 BOEHRINGER INGELHEIM PHARMACEUTICALS, INC.;BEKKALI, YOUNES;BETAGERI, RAJASHEHAR;EMMANUEL, MICHAEL, J.;HAMMACH, ABDELHAKIM;HARCKEN, HANKE, JUSTUS, JOACHIM;KIRRANE, THOMAS, MARTIN;KUZMICH, DANIEL;LEE, THOMAS, WAI-HO;LIU, PINGRONG;PATEL, USHA, R.;RAZAVI, HOSSEIN;RIETHER, DORIS;TAKAHASHI, HIDENORI;THOMSON, DAVID, S.;WANG, JI;ZINDELL, RENEE;PROUDFOOT, JOHN, ROBERT 发明人 BEKKALI, YOUNES;BETAGERI, RAJASHEHAR;EMMANUEL, MICHAEL, J.;HAMMACH, ABDELHAKIM;HARCKEN, HANKE, JUSTUS, JOACHIM;KIRRANE, THOMAS, MARTIN;KUZMICH, DANIEL;LEE, THOMAS, WAI-HO;LIU, PINGRONG;PATEL, USHA, R.;RAZAVI, HOSSEIN;RIETHER, DORIS;TAKAHASHI, HIDENORI;THOMSON, DAVID, S.;WANG, JI;ZINDELL, RENEE;PROUDFOOT, JOHN, ROBERT
分类号 A61K31/4745;A61K31/52;A61K31/5377;A61P5/44;A61P5/46;C07D209/08;C07D213/75;C07D237/20;C07D239/42;C07D307/79;C07D319/06;C07D319/08;C07D405/04;C07D405/06;C07D405/10;C07D405/14;C07D407/06;C07D471/02;C07D471/04;C07D487/04;C07D491/02;C07D491/04;C07D495/04;C07D498/02;(IPC1-7):A61K31/475 主分类号 A61K31/4745
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