发明名称 TRISUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS MODULATORS OF METABOLISM AND THE PROPHYLAXIS AND TREATMENT OF DISORDERS RELATED THERETO
摘要 The present invention relates to certain trisubstituted aryl and heteroaryl derivatives of Formula (I) that are modulators of metabolism. Accordingly, compounds of the present invention are useful in the prophylaxis or treatment of metabolic disorders and complications thereof, such as, diabetes and obesity.
申请公布号 WO2005007647(A9) 申请公布日期 2005.04.07
申请号 WO2004US22327 申请日期 2004.07.09
申请人 ARENA PHARMACEUTICALS, INC.;JONES, ROBERT, M.;SEMPLE, GRAEME;XIONG, YIFENG;SHIN, YOUNG-JUN;REN, ALBERT, S.;CALDERON, IMELDA;CHOI, JIN, SUN, KAROLINE;FIORAVANTI, BEATRIZ;LEHMANN, JUERG;BRUCE, MARC, A. 发明人 JONES, ROBERT, M.;SEMPLE, GRAEME;XIONG, YIFENG;SHIN, YOUNG-JUN;REN, ALBERT, S.;CALDERON, IMELDA;CHOI, JIN, SUN, KAROLINE;FIORAVANTI, BEATRIZ;LEHMANN, JUERG;BRUCE, MARC, A.
分类号 A61K31/4439;A61K31/513;A61P3/10;C07D239/52;C07D239/54;C07D401/12;C07D401/14;C07D403/12;C07D405/14;C07D409/14;C07D413/14;C07D417/14;(IPC1-7):C07D401/12;A61K31/506;A61K31/537;A61K31/505 主分类号 A61K31/4439
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