发明名称 |
CONJUGATES OF BIOLOGICALLY ACTIVE COMPOUNDS, METHODS FOR THEIR PREPARATION AND USE, FORMULATION AND PHARMACEUTICAL APPLICATIONS THEREOF |
摘要 |
This invention features a compound of the following formula: T-(-L-C)m, T is a transportophore, L is a bond or a linker having a molecular weight up to 240 dalton, C is a non-antibiotic therapeutic agent, and m is 1, 2, 3, 4, 5, 6, 7, or 8, in which the transportophore has an immune selectivity ratio of at least 2, the transportophore is covalently bonded to the non-antibiotic therapeutic agent via the bond or the linker, and the compound has an immune selectivity ratio of at least 2. |
申请公布号 |
WO2005027828(A2) |
申请公布日期 |
2005.03.31 |
申请号 |
WO2004US26485 |
申请日期 |
2004.08.16 |
申请人 |
SYNOVO GMBH;GUTKE, HANS-JURGEN;FLOHR, CHRISTIAN;BECK, ALBERT;MARGUTTI, SIMONA;EGGERS, MARY;GUSE, JAN-HINRICH;KHOBZAOUI, MOUSSA;BURNET, MICHAEL |
发明人 |
GUTKE, HANS-JURGEN;FLOHR, CHRISTIAN;BECK, ALBERT;MARGUTTI, SIMONA;EGGERS, MARY;GUSE, JAN-HINRICH;KHOBZAOUI, MOUSSA;BURNET, MICHAEL |
分类号 |
A01N43/04;A61K;A61K47/48;A61K49/00;C07G11/00;C07H15/00;C07H17/08 |
主分类号 |
A01N43/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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