发明名称 Fremgangsmåde til fremstilling af mikropartikler omfattende et lægemiddelstof, formulering med forlænget afgivelse, octreotidpamoat og fremgangsmåde til fremstilling heraf
摘要 A sustained release formulation of a peptide drug compound, preferably a somatostatin like octreotide, e.g. as a pamoate salt. The drug compound is present in a polymeric carrier, preferably a polylactide-co-glycolide especially a poly(lactide-co-glycolide)glucose. The formulation is preferably a depot formulation in the form of a monolithic microparticle.
申请公布号 DK175849(B1) 申请公布日期 2005.03.29
申请号 DK19900001625 申请日期 1990.07.05
申请人 NOVARTIS AG 发明人 BODMER, DAVID;FONG, JONES WING;KISSEL, THOMAS;MAULDING, HAWKINS VALLIANT;NAGELE, OSKAR;PEARSON, JANE EDNA
分类号 A61K9/14;A61K9/16;A61K9/22;A61K9/26;A61K9/50;A61K9/52;A61K38/00;A61K38/04;A61K38/22;A61K38/23;A61K38/31;A61K47/34;A61P1/00;A61P1/04;A61P1/18;A61P3/10;A61P5/02;A61P29/00;A61P35/00;C07K1/02;C07K7/06;C07K7/08;C07K14/575;C07K14/585;C07K14/655 主分类号 A61K9/14
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