发明名称 |
SYNTHESIS OF 1-[4-(2-METHOXYPHENYL) PIPERAZIN-1-YL]-3-(2,6-DIOXOPIPERIDIN-1-YL) PROPANE |
摘要 |
<p>The present invention relates to syntheses of 1-[4-(2-methoxyphenyl)piperazin-1-yl]-(2,6-dioxopiperidin-1-yl)propane and its pharmaceutically acceptable salts, preferably hydrochloride having protracted uro-selective alpha1-adrenoceptor antagonistic activity. The compound holds promise for treating benign prostatic hyperplasia (BPH).</p> |
申请公布号 |
WO2005021506(A1) |
申请公布日期 |
2005.03.10 |
申请号 |
WO2003IB03609 |
申请日期 |
2003.08.28 |
申请人 |
RANBAXY LABORATORIES LIMITED;YADAV, GYAN, CHAND;SHARMA, SOMESH;SALMAN, MOHAMMAD |
发明人 |
YADAV, GYAN, CHAND;SHARMA, SOMESH;SALMAN, MOHAMMAD |
分类号 |
A61P13/08;C07D211/88;(IPC1-7):C07D211/88;A61K31/496 |
主分类号 |
A61P13/08 |
代理机构 |
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代理人 |
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地址 |
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