发明名称 SYNTHESIS OF 1-[4-(2-METHOXYPHENYL) PIPERAZIN-1-YL]-3-(2,6-DIOXOPIPERIDIN-1-YL) PROPANE
摘要 <p>The present invention relates to syntheses of 1-[4-(2-methoxyphenyl)piperazin-1-yl]-(2,6-dioxopiperidin-1-yl)propane and its pharmaceutically acceptable salts, preferably hydrochloride having protracted uro-selective alpha1-adrenoceptor antagonistic activity. The compound holds promise for treating benign prostatic hyperplasia (BPH).</p>
申请公布号 WO2005021506(A1) 申请公布日期 2005.03.10
申请号 WO2003IB03609 申请日期 2003.08.28
申请人 RANBAXY LABORATORIES LIMITED;YADAV, GYAN, CHAND;SHARMA, SOMESH;SALMAN, MOHAMMAD 发明人 YADAV, GYAN, CHAND;SHARMA, SOMESH;SALMAN, MOHAMMAD
分类号 A61P13/08;C07D211/88;(IPC1-7):C07D211/88;A61K31/496 主分类号 A61P13/08
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