发明名称 PHARMACEUTICAL COMPOSITIONS, AZO-HETEROCYCLIC COMPOUNDS AND METHOD FOR THE PRODUCTION AND USE THEREOF
摘要 The inventive pharmaceutical composition exhibits an inhibiting activity with respect to serine proteinase (Kaspaz) and comprises an active substance embodied in the form of a pharmaceutically acceptable quantity of an azo-heterocyclic compound of general formula 1, 2 and 3 or the salts thereof with pharmacologically acceptable acid, hydrate one N-oxide.
申请公布号 WO2005018531(A2) 申请公布日期 2005.03.03
申请号 WO2004RU00331 申请日期 2004.08.25
申请人 "CHEMICAL DIVERSITY RESEARCH INSTITUTE", LTD.;IVASHCHENKO, ALEXANDER VASILIEVICH;ILYIN, ALEXEY PETROVICH;KOBAK, VLADIMIR VASILIEVICH;KRAVCHENKO, DMITRI VLADIMIROVICH;KHVAT, ALEXANDER VIKTOROVICH;TKACHENKO, SERGEY YEVGENIEVICH;OKUN, ILYA MATUSOVICH 发明人 IVASHCHENKO, ALEXANDER VASILIEVICH;ILYIN, ALEXEY PETROVICH;KOBAK, VLADIMIR VASILIEVICH;KRAVCHENKO, DMITRI VLADIMIROVICH;KHVAT, ALEXANDER VIKTOROVICH;TKACHENKO, SERGEY YEVGENIEVICH;OKUN, ILYA MATUSOVICH
分类号 A61K;A61K31/404;A61K31/427;A61K31/498;A61K31/519;A61K31/52;A61K31/525;A61K31/5377;A61P9/10;A61P25/00;A61P25/18;A61P25/28;A61P31/12;A61P31/18;C07D209/34;C07D241/44;C07D401/06;C07D401/12;C07D401/14;C07D403/06;C07D405/14;C07D409/12;C07D413/12;C07D417/12;C07D417/14;C07D475/14;C07D487/04;C07D491/12;C07D513/04;C07D513/08;C07D513/14 主分类号 A61K
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