| 发明名称 |
METODO PARA PREPARAR UM AZA-MACROLIDO COM 4 ' ' (R) -NH2 |
| 摘要 |
The subject-matter of the invention is a process for the stereoselective preparation of a compound of general formula I by stereoselective displacement by a nitrogenous nucleophilic compound of the activated alcohol functional group present at this 4'' position in a corresponding derivative of formula II. |
| 申请公布号 |
PT1144428(E) |
申请公布日期 |
2005.02.28 |
| 申请号 |
PT20000900224T |
申请日期 |
2000.01.17 |
| 申请人 |
MERIAL |
发明人 |
PATRICK LEON;GILLES ODDON;DENIS PAUZE;RONAN GUEVEL;FREDERIC LHERMITTE;GAREL, LAURENT |
| 分类号 |
A61K31/70;A61P31/00;C07B61/00;C07H17/08;(IPC1-7):C07H17/08 |
主分类号 |
A61K31/70 |
| 代理机构 |
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