发明名称 Heteroaril süksinamidler ve metalloproteinaz inhibitörü olarak kullanimlari
摘要 Mevcut bulus, formül (I) bilesiklerine yöneliktir ve burada, R1, r2, R3, R4, R5, X, Y ve (Ia) burada tanimlandigi gibidir. Bu bilesikler, metaloproteinazin bulusa ait bilesiklerin etkili miktarlariyla temas ettirerek, metaloproteinaz aktivitesini inhibe etmede kullanima elverislidir.
申请公布号 TR200402157(T2) 申请公布日期 2005.02.21
申请号 TR20040002157T 申请日期 1997.10.06
申请人 AGOURON PHARMACEUTICALS, INC.;SYNTEX (U.S.A.) INC. 发明人 STEVEN L. BENDER;ARLINDO L. CASTELHANO;WESLEY K. M. CHONG;MELWYN A. ABREO;ROLAND J. BILLEDEAU;JIAN JEFFREY CHEN;JUDITH G. DEAL
分类号 C07D233/58;A61K31/00;A61K31/34;A61K31/341;A61K31/38;A61K31/381;A61K31/40;A61K31/4025;A61K31/407;A61K31/415;A61K31/4164;A61K31/4178;A61K31/44;A61K31/4427;A61K31/443;A61K31/4433;A61K31/4436;A61K31/4439;A61K31/55;A61K38/00;A61P1/00;A61P1/02;A61P9/00;A61P9/10;A61P19/00;A61P19/02;A61P19/10;A61P29/00;A61P35/00;A61P43/00;C07D207/32;C07D207/327;C07D207/337;C07D231/12;C07D233/54;C07D233/56;C07D307/54;C07D333/24;C07D333/26;C07D401/04;C07D401/10;C07D401/12;C07D401/14;C07D403/12;C07D405/10;C07D405/12;C07D405/14;C07D409/12;C07D487/04;C07D487/08;C07D498/08;C07D521/00;C07K5/072;(IPC1-7):C07D207/327;C07K5/078;A61K38/05;C07D401/00;C07D403/00;C07D405/00;C07D409/00 主分类号 C07D233/58
代理机构 代理人
主权项
地址