摘要 |
Compounds represented by Formula (I): or a pharmaceutically acceptable salt or N-oxide thereof, wherein R1 is Formula (II, III, IV, V or VI); R2 is Formula (VII, VIII, IX or X);< >and R3 is C0-4 alkyl, are useful in the treatment of cancer. |
申请人 |
OSI PHARMACEUTICALS, INC.;WYNNE, GRAHAM, MICHAEL;DOYLE, KEVIN;AHMED, SALEH;LI, AN-HU;KEILY, JOHN FRASER;RASAMISON, CHRYSTELLE;PEGG, NEIL ANTHONY;SABA, IMAAD;THOMAS, CLAIRE;SMYTH, DON;SADIQ, SHAZIA;NEWTON, GARY;DAWSON, GRAHAM;CREW, ANDREW PHILIP;CASTELANO, ARLINDO LUCAS |
发明人 |
WYNNE, GRAHAM, MICHAEL;DOYLE, KEVIN;AHMED, SALEH;LI, AN-HU;KEILY, JOHN FRASER;RASAMISON, CHRYSTELLE;PEGG, NEIL ANTHONY;SABA, IMAAD;THOMAS, CLAIRE;SMYTH, DON;SADIQ, SHAZIA;NEWTON, GARY;DAWSON, GRAHAM;CREW, ANDREW PHILIP;CASTELANO, ARLINDO LUCAS |