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发明名称
-内醯胺抑制剂中间体之合成方法(一) PROCESS FOR SYNTHESIZING -LACTAMASE INHIBITOR INTERMEDIATES
摘要
本发明系有关一种制造下式之中间体二环杂芳基-2-羧酸的制法093113267-p01.bmp(其中X和Y如说明书之定义),其可藉由将下式位置性可水解酯类之混合物093113267-p02.bmp(其中X、Y和R如说明书之定义)进行选择性水解,而用于制备β-内醯胺抑制剂。093113267-p01.bmp
申请公布号
TW200505925
申请公布日期
2005.02.16
申请号
TW093113267
申请日期
2004.05.12
申请人
惠氏控股公司
发明人
拉米契温凯玛土;马克爱德华露平
分类号
C07D487/06
主分类号
C07D487/06
代理机构
代理人
何金涂;林荣琳
主权项
地址
美国
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