发明名称 INTERMEDIATE PRODUCTS OF THE SYNTHESIS OF FLUORIZED INHIBITORS OF ASPARTIC PROTEASES
摘要 The invention relates to compounds of general formula (I) wherein R represents H or an amine-function protective group such as a benzyl group which is substituted or not, a phenyl group which is substituted or not such as paramethoxy phenyl, or a phenyl group substituted by a group of the formula CH(Ph)CH2-OCH3 (R or S).
申请公布号 WO2005012276(A2) 申请公布日期 2005.02.10
申请号 WO2004FR02049 申请日期 2004.07.30
申请人 CENTRE NATIONALE DE LA RECHERCHE SCIENTIFIQUE;UNIVERSITE DE PARIS SUD XI;BONNET-DELPON, DANIELE;BEGUE, JEAN-PIERRE;CROUSSE, BENOIT;MAGUEUR, GUILLAUME 发明人 BONNET-DELPON, DANIELE;BEGUE, JEAN-PIERRE;CROUSSE, BENOIT;MAGUEUR, GUILLAUME
分类号 A61K31/335;A61P31/18;A61P33/06;C07D303/36 主分类号 A61K31/335
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