发明名称 |
DERIVADOS DE SULFONILFENILCARBAMOIL SUSTITUIDOS DE 9-DEOXO-9-DIHIDRO-9A-AZA-9A-HOMOERTITROMICINA A Y 5-O- DESOSAMINIL-9-DEOXO-9-DIHIDRO-9A-AZA-9A-HOMOERITROMNOLIDA A, COMPOSICION FARMACEUTICA, PROCEDIMIENTO DE PREPARACION, UTIL PARA ESTERILIZAR SALAS |
摘要 |
The invention relates to substituted 9a-N-{N'-[4-(sulfonyl)phenyl]carbamoyl} derivatives of 9-deoxo-9-dihydro-9a-aza-9a-homoerithromycin A and 5-0-desosaminyl-9-deoxo-9-di-hydro-9a-aza-9a-homoerithronolide A, novel semisynthetic macrolide antibiotics of the azalide series general formula (1), wherein R represents H or cladinosyl moiety and R1 represents chloro, amino, phenylamino, 2-pyridylamino, 3,4-dimethyl-4-isoxalylamino and 5-methyl-3-isoxazolylamino group, and pharmaceutically acceptable addition salts thereof with inorganic or organic acids. to the process for their preparation of pharmaceutical composition as well as the use their compositions for sterilization rooms and medical instruments as well as for protection of wall and wooden coatings |
申请公布号 |
CL2003002294(A1) |
申请公布日期 |
2005.01.28 |
申请号 |
CL20030002294 |
申请日期 |
2003.11.10 |
申请人 |
PLIVA D.D. |
发明人 |
KUJUNDZI NEDJEIJO, BUKVIC KRAJACI MIRJANA, BRAJSAKARMEN |
分类号 |
A61K31/7048;A61P31/00;C07H17/08;(IPC1-7):A61K31/704 |
主分类号 |
A61K31/7048 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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