| 摘要 |
The invention relates to chemical compounds in the form of racemates, enantiomers and/or diastereomers of general formula (I), wherein R represent s the non-modified part of a variable pharmaceutical active substance molecule , B represents a spacer and Toc and corresponds to formula (II), R.prime., R.prime..prime. and R.prime..prime..prime. are H or methyl for tocopherol an d A is C=X, SOm, X and/or CH2. X is O, S or NR1 (n = 1) and/or S or NR1 (n = 0 ) and B is a group X-R 2 y, wherein Y is C=X, SOm or C (XR 3 ) R4, and n is 0 - 6, preferably 0,1, 2 or 3 and m represents 1 or 2. R1 represents H, C1 - C10 - alkyl, preferably C1 - C6-alkyl and/or aryl, Het or an aryl radical and/or a Het radical connected via a C1 - C6 spacer, preferably C1 - C3 and R2 is selected from the group containing alkene, arylene and/or Het spacer and combinations thereof and can be combined directly with each other or via the A radical and/or via the group XO-A-Xp, wherein o and p can be equal or different and are 0, 1 or 2, and R3 and R4 represent H, C1 - C10 alkyl, preferably C1-C6-alkyl and/or aryl, Het or an aryl radical and/or a Het radical bound by means of a C1 - C6, preferably C1 - C3 spacer.
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