发明名称 Benzimidazole derivatives, their production and use
摘要 A method for producing a compound represented by the formula:wherein the ring A is a benzene ring which may be substituted in addition to the R' group; R<1 >is hydrogen or an optionally substituted hydrocarbon residue; X is a direct bond or a spacer having an atomic length or two or less between the phenylene group and the phenyl group; Y is -O-, -S(O)m- or -N(R<4>)- wherein m is an integer of 0, 1 or 2 and R<4 >is hydrogen or an optionally substituted alkyl group; R' is carboxyl, an ester thereof, an amide thereof or a group capable of forming an anion or a group convertible thereinto; n is an integer of 1 or 2; or a salt thereof, which comprises deprotecting a compound represented by the formula:wherein R is triphenylmethyl, 2-tetrahydropyranyl, methoxymethyl or ethoxy methyl, the other symbols as defined above; or a salt thereof.
申请公布号 US6844443(B2) 申请公布日期 2005.01.18
申请号 US20030612984 申请日期 2003.07.07
申请人 发明人
分类号 A61P9/12;C07D235/02;C07D235/26;C07D235/28;C07D235/30;C07D403/10;(IPC1-7):C07D257/04 主分类号 A61P9/12
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