| 发明名称 |
CATHEPSIN CYSTEINE PROTEASE INHIBITORS, PHARMACEUTICAL COMPOSITION BASED THEREON AND A PROCESS FOR PREPARATION THEREOF |
| 摘要 |
This invention relates to a novel class of compounds that are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, such as osteoporosis.
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| 申请公布号 |
UA77768(C2) |
申请公布日期 |
2005.01.17 |
| 申请号 |
UA20041008005 |
申请日期 |
2003.02.28 |
| 申请人 |
MERCK FROSST CANADA & CO.;AXYS PHARMACEUTICALS, INC. |
发明人 |
BAYLY CHRISTOPHER I.;LI CHUNG SING;GAUTHIER JACQUES YVES;GREEN MICHAEL J;HIRSCHBEIN BERNARD L.;JANC JAMES W;PALMER JAMES T. |
| 分类号 |
A61K31/275;A61P1/02;A61P3/14;A61P19/02;A61P19/08;A61P19/10;A61P29/00;A61P35/00;C07C255/25;C07C255/46;C07C311/37;C07C317/32;C07D209/08;C07D211/26;C07D211/38;C07D213/36;C07D213/89;C07D215/12;C07D231/12;C07D233/54;C07D233/64;C07D239/06;C07D239/26;C07D241/12;C07D261/08;C07D271/06;C07D277/28;C07D295/12;C07D295/135;C07D295/22;C07D307/52;C07D333/20;C07D401/04 |
主分类号 |
A61K31/275 |
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