发明名称 Thiolactones
摘要 This invention provides new compounds, pharmaceutical compositions and diagnostic kits comprising such compounds, and methods of using such compounds for inhibiting NAALADase enzyme activity, detecting diseases where NAALADase levels are altered, inhibiting angiogenesis, effecting a TGF-beta activity or a neuronal activity, and treating a glutamate abnormality, a compulsive disorder, neuropathy, pain, a prostate disease, cancer, Huntington's disease, diabetes, a retinal disorder or glaucoma.
申请公布号 US2005004203(A1) 申请公布日期 2005.01.06
申请号 US20040791278 申请日期 2004.03.03
申请人 GUILFORD PHARMACEUTICALS INC. 发明人 SLUSHER BARBARA S.;TSUKAMOTO TAKASHI
分类号 A61K31/381;A61K31/382;A61K31/407;C07D335/02;C07D335/06;C07D495/04;C07D498/02;(IPC1-7):A61K31/407 主分类号 A61K31/381
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