摘要 |
THE INVENTION RELATES TO A NOVEL SUSTAINED RELEASE PHARMACEUTICAL FORMULATION ADAPTED FOR ADMINISTRATION BY INJECTION CONTAINING THE COMPOUND 7X-[9-(4,4,5,5,5-PENTAFLUOROPENTYLSULPHINYL) NONYL]OESTRA-1,3,5(10)-TRIENE-3,17B-DIOL, MORE PARTICULARLY TO A FORMULATION ADAPTED FOR ADMINISTRATION BY INJECTION CONTAINING TO COMPOUND 7a-[9-(4,4,5,5,5-PENTAFLUOROPENTYLSULPHINYL) NONYL] OESTRA- 1,3,5 (10)-TRIENE-3,17B-DIOL IN SOLUTION IN A RICINOLEATE VEHICLE WHICH ADDITIONALLY COMPRISES AT LEAST ONE ALCOHOL AND A NON-AQUEOUS ESTER SOLVENT WHICH IS MISCIBLE IN THE RICINOLEATE VEHICLE. |