发明名称 |
SUBSTITUTED THIOPHENES WITH ANTIBACTERIAL ACTIVITY |
摘要 |
Novel substituted thiophenes that are inhibitors of bacterial methionyl t-RNA synthetase (MRS) are disclosed. Also disclosed are method for their preparation and their use in therapy as anti-bacterial agents. |
申请公布号 |
WO2004078119(A3) |
申请公布日期 |
2004.12.29 |
申请号 |
WO2004US05930 |
申请日期 |
2004.02.27 |
申请人 |
REPLIDYNE INC;BERGE JOHN;JARVEST RICHARD;FRYDRYCH CATHERINE SIMONE VICT;GUILES JOSEPH;QIU JIAN;TARASOW THEODORE M |
发明人 |
BERGE JOHN;JARVEST RICHARD;FRYDRYCH CATHERINE SIMONE VICT;GUILES JOSEPH;QIU JIAN;TARASOW THEODORE M |
分类号 |
A61K;A61K31/415;A61K31/47;A61K31/505;C07D215/233;C07D235/22;C07D495/04 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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