发明名称 |
2-HYDROXYMETHYL-3,4,5-TRIHYDROXY-1-(4-PENTLYOXYBENZYL) PIPERIDINE AS GLUCOSYLCERAMIDE SYNTHASE (GCS) |
摘要 |
<p>The compound 3,4,5-piperidinetriol, 2-(hydroxymethyl)-1-[(4-(pentyloxy)phenyl)methyl]-, (2S,3S,4R,5S), or a pharmaceutically acceptable salt or prodrug thereof, is useful as an inhibitor of glucosylceramide synthase.</p> |
申请公布号 |
WO2004111001(A1) |
申请公布日期 |
2004.12.23 |
申请号 |
WO2004GB02450 |
申请日期 |
2004.06.09 |
申请人 |
OXFORD GLYCOSCIENCES (UK) LTD;ORCHARD, MICHAEL, GLEN;SCOPES, DAVID, IAN, CARTER |
发明人 |
ORCHARD, MICHAEL, GLEN;SCOPES, DAVID, IAN, CARTER |
分类号 |
A61P3/10;A61P35/00;C07D211/46;(IPC1-7):C07D211/46;A61K31/445 |
主分类号 |
A61P3/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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