发明名称 PROCESS FOR PREPARING HIGHLY FUNCTIONALIZED Y-BUTYROLACTAMS AND Y-AMINO ACIDS
摘要 The invention relates to a process for preparing highly functionalized gamma-butyrolactams and gamma-amino acids by reductive amination of mucohalic acid or its derivatives, and discloses a process for preparing pregabalin, a GABA analog with desirable medicinal activity.
申请公布号 KR20040106415(A) 申请公布日期 2004.12.17
申请号 KR20047017412 申请日期 2003.04.17
申请人 发明人
分类号 C07C227/22;C07D207/38;A61K31/198;A61K31/405;A61K31/4172;C07B61/00;C07C227/12;C07C229/00;C07C229/04;C07C229/06;C07C229/08;C07C229/28;C07C229/34;C07C229/38;C07D207/24;C07D209/18;C07D213/55;C07D233/66 主分类号 C07C227/22
代理机构 代理人
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