发明名称 Tetrapeptide derivative crystals
摘要 The invention provides crystals of N<2>-(N,N-dimethyl-L-valyl)-N-[(1S,2R)-2-methoxy-4-[(2S)-2-[(1R,2R)-1-methoxy-2-methyl-3-oxo-3-[(2-phenylethyl)amino]propyl]-1-pyrrolidinyl]-1-[(S)-1-methylpropyl]-4-oxobutyl]-N-methyl-L-valinamide or salts thereof which possess potent antitumor activity and methods for their preparation.
申请公布号 US2004254343(A1) 申请公布日期 2004.12.16
申请号 US20040490340 申请日期 2004.03.22
申请人 MIYAZAKI KOICHI;KEINO KATSUYUKI;KANADA ARIHIRO;MINAMI NOBUYOSHI 发明人 MIYAZAKI KOICHI;KEINO KATSUYUKI;KANADA ARIHIRO;MINAMI NOBUYOSHI
分类号 A61K38/00;A61P35/00;C07K5/02;C07K5/103;(IPC1-7):A61K38/06;C07K7/06 主分类号 A61K38/00
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