发明名称 PYPERAZINYL, PYPERIDINYL AND MORPHOLINYL DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS
摘要 This invention comprises the novel compounds of formula (I) wherein t, R1, R2, L, Q, X, Y, Z, and (a) have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 UA77264(C2) 申请公布日期 2004.12.15
申请号 UA20040907277 申请日期 2003.03.11
申请人 JANSSEN PHARMACEUTICA N.V. 发明人
分类号 A61K31/40;A61K31/438;A61K31/445;A61K31/454;A61K31/472;A61K31/495;A61K31/496;A61K31/506;A61K31/517;A61K31/537;A61K31/55;A61K31/551;A61K45/00;A61P1/04;A61P3/10;A61P5/00;A61P9/00;A61P9/02;A61P9/08;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/08;A61P13/10;A61P13/12;A61P15/00;A61P17/00;A61P17/04;A61P17/06;A61P17/10;A61P17/14;A61P17/16;A61P19/02;A61P19/06;A61P21/04;A61P25/00;A61P25/16;A61P25/28;A61P27/02;A61P27/06;A61P29/00;A61P31/18;A61P35/00;A61P35/02;A61P37/02;A61P37/04;A61P37/06;A61P37/08;A61P43/00;C07D207/09;C07D207/14;C07D211/26;C07D211/58;C07D213/74;C07D213/78;C07D217/02;C07D217/04;C07D239/42;C07D241/04;C07D249/12;C07D295/14;C07D295/155;C07D295/20;C07D295/22;C07D295/26;C07D307/68;C07D317/58;C07D401/04;C07D401/06;C07D401/12;C07D401/14;C07D403/04;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D413/04;C07D413/12;C07D471/10;C12Q1/48 主分类号 A61K31/40
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