发明名称 SMALL MOLECULE ENTRY INHIBITORS.
摘要 <p>The present invention concerns a compound having the formula (I) a N-oxide form, a stereochemical isomer, racemic mixture, salt prodrug, ester or metabolite thereof. It further relates to processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors with anti-retroviral agents. It further relates to their use in assays as reference compounds or as reagents. The compounds of the present invention are useful for preventing or treating infection by HIV and for treating AIDS.</p>
申请公布号 MXPA04008926(A) 申请公布日期 2004.12.13
申请号 MX2004PA08926 申请日期 2003.03.11
申请人 TIBOTEC PHARMACEUTICALS LTD. 发明人 EISSENSTAT, MICHAEL
分类号 C07D295/22;A61K31/167;A61K31/196;A61K31/27;A61K31/34;A61K31/381;A61K31/455;A61K31/5375;A61P31/18;A61P43/00;C07C229/56;C07C229/58;C07C233/55;C07C233/81;C07C235/24;C07C235/38;C07C235/56;C07C235/84;C07C237/42;C07C255/57;C07C311/21;C07C311/29;C07C311/46;C07C317/14;C07C323/56;C07D209/48;C07D209/76;C07D209/78;C07D213/56;C07D213/81;C07D213/82;C07D295/26;C07D307/68;C07D333/38;(IPC1-7):A61K31/167 主分类号 C07D295/22
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