发明名称 PROCESS FOR THE SYNTHESIS OF DISTAMYCIN AND DERIVATIVES THEREOF USING 1-METHYL-4-FORMYLAMINO-2-PYRROLECARBONYL CHLORIDE ITERATIVELY AS AN INTERMEDIATE
摘要 <p>A process for the total synthesis of Distamycin, and synthetic poly-(4 aminopyrrole -2-carboxamide) congeners thereof, using 1-methyl-4­- forinylamino-2-pyrrolecarbonyl chloride iteratively as an intermediate, is provided. The process finds application for both in solution and solid support synthetic technologies.</p>
申请公布号 WO2004106301(A1) 申请公布日期 2004.12.09
申请号 WO2004EP05821 申请日期 2004.05.28
申请人 NAXOSPHARMA S.R.L.;LOMBARDI, PAOLO 发明人 LOMBARDI, PAOLO
分类号 C07D207/34;(IPC1-7):C07D207/34 主分类号 C07D207/34
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