发明名称 |
PROCESS FOR THE SYNTHESIS OF DISTAMYCIN AND DERIVATIVES THEREOF USING 1-METHYL-4-FORMYLAMINO-2-PYRROLECARBONYL CHLORIDE ITERATIVELY AS AN INTERMEDIATE |
摘要 |
<p>A process for the total synthesis of Distamycin, and synthetic poly-(4 aminopyrrole -2-carboxamide) congeners thereof, using 1-methyl-4- forinylamino-2-pyrrolecarbonyl chloride iteratively as an intermediate, is provided. The process finds application for both in solution and solid support synthetic technologies.</p> |
申请公布号 |
WO2004106301(A1) |
申请公布日期 |
2004.12.09 |
申请号 |
WO2004EP05821 |
申请日期 |
2004.05.28 |
申请人 |
NAXOSPHARMA S.R.L.;LOMBARDI, PAOLO |
发明人 |
LOMBARDI, PAOLO |
分类号 |
C07D207/34;(IPC1-7):C07D207/34 |
主分类号 |
C07D207/34 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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