发明名称 |
CYCLICAMINO-PHENYL SULFAMATE DERIVATIVES |
摘要 |
A cyclic aminophenyl sulfamate derivative represented by the formula (I) (wherein R1 and R2 each represents hydrogen or lower alkyl; R3 and R4 each represents hydrogen, halogeno, cyano, etc.; A represents nitrogen or CH; B represents CH2, SO2, CO, optionally substituted phenyl, etc.; and R5 represents alkyl, phenyl, amino, etc.), or a salt thereof. The derivative ha s excellent steroid sulfatase inhibitory activity and is useful for the prevention of or treatments for diseases in which steroids such as estrogen and androgen participate.
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申请公布号 |
CA2526540(A1) |
申请公布日期 |
2004.12.02 |
申请号 |
CA20042526540 |
申请日期 |
2004.05.07 |
申请人 |
ASKA PHARMACEUTICAL CO., LTD. |
发明人 |
NAKAGAWA, TAKAYOSHI;FUJII, TOMOHITO;KOIZUMI, NAOYUKI;OKADA, MAKOTO;TAKEGAWA, SHIGEHIRO;IWASHITA, SHIGEKI |
分类号 |
C07D211/14;A61K31/451;A61K31/4545;A61K31/495;A61P15/00;A61P17/00;A61P25/28;A61P35/00;A61P37/06;A61P43/00;C07D211/62;C07D211/70;C07D295/08;C07D295/18;C07D295/22 |
主分类号 |
C07D211/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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