发明名称 PROCESS FOR SYNTHESIZING beta-LACTAMASE INHIBITOR IN INTERMEDIATES
摘要 There is provided a process for the preparation of bicyclicheteroaryl carboxaldehydes having the structural Formula I where X and Y are defined in the specification. The bicyclic heteroaryl carboxaldehydes are useful as intermediates in the preparation of beta-lactamase inhibitors.
申请公布号 WO2004104006(A2) 申请公布日期 2004.12.02
申请号 WO2004US14834 申请日期 2004.05.12
申请人 WYETH HOLDINGS CORPORATION;WINKLEY, MICHAEL, WILLIAM;CHAN, ANITA WAI-YIN;JIRKOVSKY, IVO, L.;KREMER, KENNETH, ALFRED, MARTIN;ZELDIS, JOSEPH;NIKITENKO, ANTONINA, ARISTOTELEVNA;STRONG, HENRY, LEE;MANSOUR, TAREK, SUHAYL;KHAFIZOVA, GULNAZ;VENKATESAN, ARANAPAKAM, MUDUMBAI 发明人 WINKLEY, MICHAEL, WILLIAM;CHAN, ANITA WAI-YIN;JIRKOVSKY, IVO, L.;KREMER, KENNETH, ALFRED, MARTIN;ZELDIS, JOSEPH;NIKITENKO, ANTONINA, ARISTOTELEVNA;STRONG, HENRY, LEE;MANSOUR, TAREK, SUHAYL;KHAFIZOVA, GULNAZ;VENKATESAN, ARANAPAKAM, MUDUMBAI
分类号 C07D487/04;C07D513/12 主分类号 C07D487/04
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