发明名称 PROCESS FOR PRODUCING PYRROLIDINE DERIVATIVE
摘要 <p>A process for industrially advantageously producing a 1,4-trans-cyclohexanecarboxylic acid derivative (1) which has excellent VLA-4 inhibitory activity and is safe; and an intermediate advantageous for the production process. The process comprises converting a compound represented by the formula (I) into a compound represented by the formula (VI) according to the following scheme.</p>
申请公布号 WO2004099136(A1) 申请公布日期 2004.11.18
申请号 WO2004JP06471 申请日期 2004.05.07
申请人 YONEDA, YOSHIYUKI;DAIICHI PHARMACEUTICAL CO., LTD.;NAKAYAMA, ATSUSHI;MACHINAGA, NOBUO;SETOGUCHI, MASAKI 发明人 NAKAYAMA, ATSUSHI;MACHINAGA, NOBUO;YONEDA, YOSHIYUKI;SETOGUCHI, MASAKI
分类号 C07D207/12;(IPC1-7):C07D207/04;C07D403/12 主分类号 C07D207/12
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