发明名称 N-BIPHENYLMETHYL AMINOCYCLOALKANECARBOXAMIDE DERIVATIVES WITH A SUBSTIITUENT ON THE METHYL USEFUL AS BRADYKININ ANTAGONISTS.
摘要 <p>N-Biphenyl(substituted methyl)aminocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.</p>
申请公布号 MXPA04007660(A) 申请公布日期 2004.11.10
申请号 MX2004PA07660 申请日期 2003.02.04
申请人 MERCK & CO., INC. 发明人 WAI. JENNY MIU-CHUN
分类号 A61K31/166;A61K31/24;A61K31/41;A61K31/42;A61K31/4245;A61K31/505;A61P1/02;A61P1/04;A61P1/16;A61P1/18;A61P9/10;A61P11/00;A61P11/06;A61P11/08;A61P13/10;A61P13/12;A61P17/02;A61P17/06;A61P19/02;A61P19/08;A61P21/00;A61P25/04;A61P25/06;A61P25/28;A61P27/16;A61P29/00;A61P31/04;A61P35/00;A61P37/08;C07C237/24;C07D213/82;C07D239/28;C07D257/04;C07D261/18;C07D271/06;C07D403/12;C07D413/12;(IPC1-7):C07C237/24;C07D271/00;C07D261/00;C07D239/00 主分类号 A61K31/166
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