发明名称 |
N-BIPHENYLMETHYL AMINOCYCLOALKANECARBOXAMIDE DERIVATIVES WITH A SUBSTIITUENT ON THE METHYL USEFUL AS BRADYKININ ANTAGONISTS. |
摘要 |
<p>N-Biphenyl(substituted methyl)aminocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.</p> |
申请公布号 |
MXPA04007660(A) |
申请公布日期 |
2004.11.10 |
申请号 |
MX2004PA07660 |
申请日期 |
2003.02.04 |
申请人 |
MERCK & CO., INC. |
发明人 |
WAI. JENNY MIU-CHUN |
分类号 |
A61K31/166;A61K31/24;A61K31/41;A61K31/42;A61K31/4245;A61K31/505;A61P1/02;A61P1/04;A61P1/16;A61P1/18;A61P9/10;A61P11/00;A61P11/06;A61P11/08;A61P13/10;A61P13/12;A61P17/02;A61P17/06;A61P19/02;A61P19/08;A61P21/00;A61P25/04;A61P25/06;A61P25/28;A61P27/16;A61P29/00;A61P31/04;A61P35/00;A61P37/08;C07C237/24;C07D213/82;C07D239/28;C07D257/04;C07D261/18;C07D271/06;C07D403/12;C07D413/12;(IPC1-7):C07C237/24;C07D271/00;C07D261/00;C07D239/00 |
主分类号 |
A61K31/166 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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