发明名称 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
摘要 Compounds having kappa opioid agonist activity, compositions containing them and method of using them as analgesics and pruritic agents are provided. The compounds of formulae I, II, III and IV have the structure: wherein X, X4, X5, X7, X9; R1, R2, R3, R4; and Y, Z and n are as described in the specification
申请公布号 US2004220112(A1) 申请公布日期 2004.11.04
申请号 US20030455687 申请日期 2003.06.05
申请人 KRUSE LAWRENCE I.;CHANG AN-CHIH;DEHAVEN-HUDKINS DIANE L.;FARRAR JOHN J.;GAUL FORREST;KUMAR VIRENDRA;MARELLA MICHAEL ANTHONY;MAYCOCK ALAN L.;ZHANG WEI YUAN 发明人 KRUSE LAWRENCE I.;CHANG AN-CHIH;DEHAVEN-HUDKINS DIANE L.;FARRAR JOHN J.;GAUL FORREST;KUMAR VIRENDRA;MARELLA MICHAEL ANTHONY;MAYCOCK ALAN L.;ZHANG WEI YUAN
分类号 C07D295/12;A61K31/40;A61K31/404;A61K31/405;A61K31/4427;A61K31/4439;A61K31/495;A61K31/496;A61P17/04;A61P25/04;C07D207/09;C07D207/12;C07D209/08;C07D209/18;C07D209/42;C07D213/56;C07D241/04;C07D273/08;C07D401/12;C07D403/06;C07D403/12;(IPC1-7):A61K38/04;A61K31/675;A61K31/401 主分类号 C07D295/12
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