发明名称 SYNTHESIS OF 2-HYDROXY-N,N-DIMETHYL-3-[[2-[1(R)-(5-METHYL-2-FURANYL)PROPYL]AMINO]-3,4-DIOXO-1-CYCLOBUTEN-1-YL]AMINO]BENZAMIDE
摘要 Disclosed is a process for making the compound of formula (I), using the compounds of formulas (II), (Q), and (XI) or (XII) (II), wherein A is select ed from the group consisting of Br, Cl and (I) (with Br being preferred); and R represents (C1-C10)alkyl. Also disclosed are intermediate compounds that are made in the disclosed process.
申请公布号 CA2522748(A1) 申请公布日期 2004.11.04
申请号 CA20042522748 申请日期 2004.04.16
申请人 SCHERING CORPORATION 发明人 SUDHAKAR, ANANTHA;WINTERS, JASON L.;KIM-MEADE, AGNES S.;ZHANG, SHUYI;MCALLISTER, TIMOTHY L.;YIN, JIANGUO;SCHUMACHER, DORIS P.;FU, XIAOYONG
分类号 C07C235/60;C07D307/52;(IPC1-7):C07D307/52;C07C205/60 主分类号 C07C235/60
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