发明名称 CYCLIC AMINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF INFLAMMATION-RELATED DISORDERS MEDIATED BY BRADYKININ
摘要 <p>Compounds of formula (I) are effective for treatment of pain and diseases, such as inflammation mediated diseases. The invention encompasses novel compounds, pharmaceutically acceptable derivatives thereof, pharmaceutical compositions and methods for prophylaxis and treatment of diseases and other maladies or conditions involving pain, inflammation mediated by Bradykinin. The subject invention also relates to processes for making such compounds as well as to intermediates useful in such processes wherein q, t, R, R&lt;a&gt;, R&lt;b&gt;, R&lt;c&gt; and R&lt;2&gt; are as defined herein.</p>
申请公布号 WO2004092164(A1) 申请公布日期 2004.10.28
申请号 WO2004US11670 申请日期 2004.04.12
申请人 AMGEN, INC.;ARRAY BIOPHARMA, INC.;GRONEBERG, ROBERT, D.;ZHAN, JAMES;ASKEW, BEN;D'AMICO, DERIN;HAN, NIANH;FOTSCH, CHRISTOPHER, H.;LIU, QINGLAN;RIAHI, BABAK;ZHU, JIAWANG;YANG, KEVIN;CHEN, JIAN, J.;NOMAK, RANA 发明人 GRONEBERG, ROBERT, D.;ZHAN, JAMES;ASKEW, BEN;D'AMICO, DERIN;HAN, NIANH;FOTSCH, CHRISTOPHER, H.;LIU, QINGLAN;RIAHI, BABAK;ZHU, JIAWANG;YANG, KEVIN;CHEN, JIAN, J.;NOMAK, RANA
分类号 A61K31/425;A61K31/4523;A61K31/454;A61K31/4545;A61K31/4709;A61K31/517;A61K31/55;A61P29/00;C07D207/48;C07D211/96;C07D215/58;C07D217/22;C07D401/12;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/02;C07D413/14;C07D417/02;C07D417/12;C07D417/14;(IPC1-7):C07D405/12;A61K31/452 主分类号 A61K31/425
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