发明名称 11-PHENYL-DIBENZODIAZEPINE DERIVATIVES AS RXR-ANTAGONISTS
摘要 The present invention relates to novel benzodiazepine compounds exhibiting R XR- antagonist efficacy, for delaying progression of, preventing or treating a condition or disease being associated with RXR-antagonism, in particular selected from diabetes, complication of diabetes such as retinopathy, nephropathy, neuropathy, and hyperlipidemia, obesity, dyslipidemia, and osteoporosis.
申请公布号 CA2521337(A1) 申请公布日期 2004.10.21
申请号 CA20042521337 申请日期 2004.04.08
申请人 NOVARTIS AG 发明人 UCHIYAMA, HIDEFUMI;MITANI, HIRONOBU;SAKAKI, JUNICHI;KONISHI, KAZUHIDE;KISHIDA, MASASHI;KIMURA, MASAAKI
分类号 A61P3/00;C07D243/10;C07D243/38;(IPC1-7):C07D243/38;A61K31/551 主分类号 A61P3/00
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