发明名称 Efficient process for the preparation of a factor Xa inhibitor
摘要 The present invention relates to the process for the preparation of the compound of Formula I: from its corresponding 3-cyano-4-fluorophenyl-pyrazole and intermediates useful therein.
申请公布号 US2004198787(A1) 申请公布日期 2004.10.07
申请号 US20040826099 申请日期 2004.04.15
申请人 LI HUI-YIN;ANZALONE LUIGI;JIN FUQIANG;MELONI DAVID J.;SUN JUNG-HUI;ROSSANO LUCIUS T.;TELEHA CHRISTOPHER A.;ZHOU JIACHENG;SMYSER THOMAS E. 发明人 LI HUI-YIN;ANZALONE LUIGI;JIN FUQIANG;MELONI DAVID J.;SUN JUNG-HUI;ROSSANO LUCIUS T.;TELEHA CHRISTOPHER A.;ZHOU JIACHENG;SMYSER THOMAS E.
分类号 C07D231/14;A61K;A61K31/4178;A61K31/42;A61K31/422;A61K31/423;A61P;A61P7/02;C07C51/41;C07C57/145;C07D;C07D403/12;C07D413/14;(IPC1-7):A61K31/42 主分类号 C07D231/14
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