发明名称 |
Cyclohept'b!indole derivatives as spla2 inhibitors |
摘要 |
A novel class of tricyclic compounds of the following formula (1): (formula I); is disclosed together with the use of such compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of inflammatory diseases such as septic shock.
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申请公布号 |
US2004198801(A1) |
申请公布日期 |
2004.10.07 |
申请号 |
US20040483939 |
申请日期 |
2004.01.15 |
申请人 |
KINNICK MICHAEL DEAN;MIHELICH EDWARD DAVID;MORIN JOHN MICHAEL;SALL DANIEL JON;SAWYER JASON SCOTT |
发明人 |
KINNICK MICHAEL DEAN;MIHELICH EDWARD DAVID;MORIN JOHN MICHAEL;SALL DANIEL JON;SAWYER JASON SCOTT |
分类号 |
A61K31/403;A61P1/00;A61P11/00;A61P19/00;A61P29/00;A61P31/00;A61P43/00;C07D209/94;(IPC1-7):C07D209/56 |
主分类号 |
A61K31/403 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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